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Tirzepetide

Tirzepatide is a cutting-edge research peptide designed to activate both GIP and GLP-1 receptors—two key regulators of insulin and glucose metabolism. By mimicking the body’s natural incretin hormones, Tirzepatide enhances insulin secretion, improves insulin sensitivity, and helps regulate appetite and body weight.

It has gained significant attention in the scientific community for its potential role in addressing metabolic disorders such as type 2 diabetes, obesity, and non-alcoholic fatty liver disease. Research models have shown impressive reductions in blood glucose levels and sustained weight loss, often outperforming GLP-1 agonists alone.

Tirzepatide is being actively investigated for its multi-pathway benefits, including effects on cardiovascular health and inflammatory markers. While promising, it remains strictly for laboratory research use and is not approved for human consumption or clinical therapy. For qualified professionals exploring metabolic modulation, Tirzepatide represents a powerful tool in advancing understanding of dual incretin mechanisms.

Peptides will arrive in a lyophilized (powder) form for maximum stability

$124.97

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🧬 Overview

Tirzepatide is a synthetic 39-amino acid peptide that functions as a dual agonist of glucose-dependent insulinotropic polypeptide (GIP) and glucagon-like peptide-1 (GLP-1) receptors. Originally developed for metabolic research, it has become a focus of preclinical investigations into peptide-based regulation of glycemic control, insulin response, and energy metabolism. Tirzepatide is currently under patent protection and has been studied extensively in rodent and non-human primate models related to glucose modulation and pancreatic function.

⚙️ Mechanism of Action

As a dual incretin receptor agonist, Tirzepatide interacts with both the GIP and GLP-1 pathways, which play key roles in postprandial glucose homeostasis. In preclinical animal models, it has been observed to influence insulin secretion, delay gastric emptying, and modulate glucagon levels. These effects have made it a peptide of interest in laboratory studies examining metabolic feedback systems, endocrine signaling, and pancreatic islet cell responsiveness under hyperglycemic conditions.

🧪 Key Research Focus Areas

Rodent and primate studies using Tirzepatide have explored its impact on body mass regulation, insulin sensitivity, lipid profiles, and hepatic glucose production. Additional investigations have assessed its potential in regulating satiety signaling, gut hormone expression, and nutrient absorption pathways. Researchers continue to explore its application in models simulating metabolic dysregulation, beta-cell stress, and incretin resistance.

⏳ Extended Research Interest

In addition to short-term studies on glycemic markers, long-term preclinical trials have examined Tirzepatide’s effects on cardiovascular biomarkers, inflammatory cytokines, and adipose tissue remodeling in animal models. Some research has also investigated its interaction with neuroendocrine circuits involved in feeding behavior and hypothalamic signaling, though human research remains proprietary and limited to clinical development channels.

🧫 Safety & Tolerability (Research Use Only)

In laboratory models, Tirzepatide has generally shown a favorable research profile with a well-characterized pharmacokinetic and pharmacodynamic footprint. However, this compound is under active patent protection and is not approved for human or veterinary use. It is intended strictly for scientific research and in vitro experimentation. All research must comply with institutional, legal, and ethical standards regarding the use of synthetic peptides.

🧬 Sequencing & Structural Data

  • Sequence: H-Aib-Gly-Glu-Gly-Thr-Phe-Thr-Ser-Asp-Val-Ser-Ser-Tyr-Leu-Glu-Gly-Gln-Ala-Ala-Lys-Glu-Phe-Ile-Ala-Trp-Leu-Val-Lys-Gly-Arg-Gly-Asp-Phe-Tyr-Glu-Ile-Gln-Gln-Ala-Lys-NH₂
  • Molecular Formula: C225H348N48O68
  • Molecular Weight: 4813.45 g/mol
  • CAS Number: 2023788-19-2
  • PubChem CID: 145996610
  • Synonyms: LY3298176, Tirzepatide Acetate

📚 References

  1. https://pubmed.ncbi.nlm.nih.gov/32898345/
  2. https://pubmed.ncbi.nlm.nih.gov/32152636/
  3. https://pubmed.ncbi.nlm.nih.gov/30526886/
  4. https://pubmed.ncbi.nlm.nih.gov/31161971/
  5. https://pubmed.ncbi.nlm.nih.gov/34476770/

⚠️ Legal Disclaimer

ALL ARTICLES AND PRODUCT INFORMATION PROVIDED ON THIS WEBSITE ARE FOR INFORMATIONAL AND EDUCATIONAL PURPOSES ONLY.

The products offered on this website are furnished for in-vitro laboratory research only. In-vitro studies (Latin: “in glass”) are performed outside of living organisms. These products are not medicines or drugs, and they have not been approved by the FDA to prevent, treat, or cure any medical condition, ailment, or disease. Under no circumstances should these products be introduced into the human or animal body, whether by injection, ingestion, topical application, or any other route. Bodily introduction is strictly prohibited by law.

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